Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50008054
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515269(CHEMBL4462592)
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50032750(CHEMBL3355181)
Affinity DataIC50: 206nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515263(CHEMBL4531109)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50032750(CHEMBL3355181)
Affinity DataIC50: 311nMAssay Description:Inhibition of human JNK2alpha2 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515266(CHEMBL4531954)
Affinity DataIC50: 350nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515263(CHEMBL4531109)
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant human EGFR T790M/L858R double mutant (696 to end residues) using GGMEDIYFEFMGGKKK as substrate measured after 40 mins in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515271(CHEMBL4551217)
Affinity DataIC50: 590nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515270(CHEMBL4464624)
Affinity DataIC50: 620nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515269(CHEMBL4462592)
Affinity DataIC50: 710nMAssay Description:Inhibition of human JNK2alpha2 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515272(CHEMBL4442806)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515269(CHEMBL4462592)
Affinity DataIC50: 820nMAssay Description:Inhibition of human JNK1alpha1 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515260(CHEMBL4451516)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515267(CHEMBL4470329)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515268(CHEMBL4483382)
Affinity DataIC50: 2.37E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515275(CHEMBL4579302)
Affinity DataIC50: 2.43E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515264(CHEMBL4533188)
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515263(CHEMBL4531109)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human EGFR L858R mutant (696 to end residues) using poly (Glu, Tyr) 4:1 as substrate measured after 40 mins in presence of [gamma33P]AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515265(CHEMBL1213862)
Affinity DataIC50: 6.57E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515262(CHEMBL4449405)
Affinity DataIC50: 7.65E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase Yes(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of recombinant human full-length yes using poly(Glu, Tyr) 4:1 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of recombinant human Abl Q252H mutant (27 to end residues) using EAIYAAPFAKKK as substrate measured after 40 mins in presence of [gamma33P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515261(CHEMBL4560317)
Affinity DataIC50: 8.89E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515273(CHEMBL4483514)
Affinity DataIC50: 9.76E+3nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50032750(CHEMBL3355181)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human JNK1alpha1 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human Abl Y253F mutant (27 to end residues) using EAIYAAPFAKKK as substrate measured after 40 mins in presence of [gamma33P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 1.39E+4nMAssay Description:Inhibition of recombinant human Abl (27 to end residues) using EAIYAAPFAKKK as substrate measured after 40 mins in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515274(CHEMBL4461363)
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of recombinant human full-length JNK3 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515270(CHEMBL4464624)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK1alpha1 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK2alpha2 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515271(CHEMBL4551217)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK2alpha2 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515259(CHEMBL4470981)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK1alpha1 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515270(CHEMBL4464624)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK2alpha2 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515263(CHEMBL4531109)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK2alpha2 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515271(CHEMBL4551217)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK1alpha1 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandPNGBDBM50515263(CHEMBL4531109)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK1alpha1 using ATF2 as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed