Compile Data Set for Download or QSAR
Report error Found 197 Enz. Inhib. hit(s) with all data for entry = 50008215
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516776(CHEMBL4437741)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516789(CHEMBL4559193)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516782(CHEMBL4592199)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516789(CHEMBL4559193)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516776(CHEMBL4437741)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516789(CHEMBL4559193)
Affinity DataEC50:  13nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516797(CHEMBL4576974)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516776(CHEMBL4437741)
Affinity DataEC50:  26nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataEC50:  41nMAssay Description:Antagonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516776(CHEMBL4437741)
Affinity DataEC50:  57nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516789(CHEMBL4559193)
Affinity DataEC50:  68nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516787(CHEMBL4556046)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516789(CHEMBL4559193)
Affinity DataEC50:  126nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516782(CHEMBL4592199)
Affinity DataEC50:  129nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516788(CHEMBL4483617)
Affinity DataKi:  272nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516803(CHEMBL4450995)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516782(CHEMBL4592199)
Affinity DataEC50:  306nMAssay Description:Agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as inhibition of NKH477-stimulated intracellular cAMP levels after 30 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516798(CHEMBL4579868)
Affinity DataKi:  395nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516801(CHEMBL4451793)
Affinity DataEC50:  437nMAssay Description:Antagonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516793(CHEMBL4450401)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516782(CHEMBL4592199)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516803(CHEMBL4450995)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516775(CHEMBL3596703)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516801(CHEMBL4451793)
Affinity DataEC50:  1.17E+3nMAssay Description:Antagonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516780(CHEMBL4462864)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516784(CHEMBL4441442)
Affinity DataKi:  1.32E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50200170(SR-144528 | 5-(4-chloro-3-methylphenyl)-1-(4-methy...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516790(CHEMBL4470152)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516776(CHEMBL4437741)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516783(CHEMBL4446746)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516797(CHEMBL4576974)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516791(CHEMBL4451217)
Affinity DataKi:  2.86E+3nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516775(CHEMBL3596703)
Affinity DataEC50:  3.31E+3nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516798(CHEMBL4579868)
Affinity DataEC50:  3.98E+3nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB2 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516774(CHEMBL4587737)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516786(CHEMBL4459664)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516797(CHEMBL4576974)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516792(CHEMBL4445661)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516788(CHEMBL4483617)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516781(CHEMBL4468254)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516780(CHEMBL4462864)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516800(CHEMBL4533663)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516804(CHEMBL4519212)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516796(CHEMBL4550200)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516786(CHEMBL4459664)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516787(CHEMBL4556046)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516802(CHEMBL1385951)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50516784(CHEMBL4441442)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB2R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
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