Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50008076
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50515480(CHEMBL4436879)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50456168(CHEMBL1800685)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50515476(CHEMBL4577585)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50515477(CHEMBL4538561)
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50515478(CHEMBL4455311)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50515475(CHEMBL4458922)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetP2Y purinoceptor 14(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50515479(CHEMBL4526840)
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at human P2Y14R stably expressed in human forskolin treated THP1 cells assessed as reduction in P2Y14R agonist UDPG-induced inhib...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed