Compile Data Set for Download or QSAR
Report error Found 138 Enz. Inhib. hit(s) with all data for entry = 50009606
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530438(Mosapramine | Mosapramine hydrochloride)
Affinity DataKi:  0.0300nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530438(Mosapramine | Mosapramine hydrochloride)
Affinity DataKi:  0.0300nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50397999(CHEMBL2180796)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50530441(CHEMBL4448109)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50530441(CHEMBL4448109)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50397999(CHEMBL2180796)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274351(2-(6,8-Dichloro-2-(4-nitrophenyl)imidazo[1,2-a]pyr...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274351(2-(6,8-Dichloro-2-(4-nitrophenyl)imidazo[1,2-a]pyr...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Palack£

Curated by ChEMBL
LigandPNGBDBM50247053(Tiprolisant | 1-(3-(3-(4-chlorophenyl)propoxy)prop...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
Palack£

Curated by ChEMBL
LigandPNGBDBM50247053(Tiprolisant | 1-(3-(3-(4-chlorophenyl)propoxy)prop...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of Guinea Pig Ileum H3RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189854(6-bromo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  0.25nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189841(6-iodo-2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]...)
Affinity DataKi:  0.330nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50060095(2-[6,8-Dichloro-2-(4-chloro-phenyl)-imidazo[1,2-a]...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50060095(2-[6,8-Dichloro-2-(4-chloro-phenyl)-imidazo[1,2-a]...)
Affinity DataKi:  0.410nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530421(CHEMBL4585201)
Affinity DataKi:  0.5nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530421(CHEMBL4585201)
Affinity DataKi:  0.5nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274258(2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...)
Affinity DataKi:  0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274258(2-(6,8-Dichloro-2-(4-methoxyphenyl)imidazo[1,2-a]p...)
Affinity DataKi:  0.537nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530440(CHEMBL4548796)
Affinity DataKi:  0.75nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530440(CHEMBL4548796)
Affinity DataKi:  0.75nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274561(4-(2-(4-Chlorophenyl)-3-(2-(dipropylamino)-2-oxoet...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274561(4-(2-(4-Chlorophenyl)-3-(2-(dipropylamino)-2-oxoet...)
Affinity DataKi:  0.860nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274259(N-Butyl-2-(6,8-dichloro-2-(4-methoxyphenyl)imidazo...)
Affinity DataKi:  0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50274259(N-Butyl-2-(6,8-dichloro-2-(4-methoxyphenyl)imidazo...)
Affinity DataKi:  0.882nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189848(2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imid...)
Affinity DataKi:  0.990nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189848(2-[4-(3,4-dichlorophenyl)piperazin-1-ylmethyl]imid...)
Affinity DataKi:  0.990nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50408728(CHEMBL339816)
Affinity DataKi:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50408728(CHEMBL339816)
Affinity DataKi:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50120543(7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  2nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50386935(CHEMBL2048680)
Affinity DataIC50: 2nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50386935(CHEMBL2048680)
Affinity DataIC50: 2nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50120543(7-Methyl-2-[4-(3-piperidin-1-yl-propoxy)-phenyl]-i...)
Affinity DataKi:  2nMAssay Description:Inhibition of H3R (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530439(CHEMBL4456416)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50530442(CHEMBL4461114)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530439(CHEMBL4456416)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50530442(CHEMBL4461114)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human PDE10More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50530425(CHEMBL4454665)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of FLAG-tagged human PDE4B2 expressed in Escherichia coli cells after 20 mins in presence of [3H]-cAMP by top count analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
LigandPNGBDBM50530425(CHEMBL4454665)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of FLAG-tagged human PDE4B2 expressed in Escherichia coli cells after 20 mins in presence of [3H]-cAMP by top count analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataKi:  2.80nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50189845(2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo...)
Affinity DataKi:  2.80nMAssay Description:Agonist activity at dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50386917(CHEMBL2048662)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530427(CHEMBL4562585)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50530427(CHEMBL4562585)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50386917(CHEMBL2048662)
Affinity DataIC50: 3nMAssay Description:Inhibition of GSK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetTranslocator protein(Human)
Palack£

Curated by ChEMBL
LigandPNGBDBM50045880(2-[5-Chloro-2-(4-chloro-phenyl)-1H-indol-3-yl]-N,N...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
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