Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50008245
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517072(CHEMBL4450922)
Affinity DataEC50:  940nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517072(CHEMBL4450922)
Affinity DataEC50:  230nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517073(CHEMBL4434980)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517074(CHEMBL1905057)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517075(CHEMBL4560492)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517076(CHEMBL4593957)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517077(CHEMBL4452828)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517074(CHEMBL1905057)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517075(CHEMBL4560492)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517078(CHEMBL4556197)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517076(CHEMBL4593957)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517077(CHEMBL4452828)
Affinity DataEC50:  5.53E+3nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517078(CHEMBL4556197)
Affinity DataEC50:  992nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517073(CHEMBL4434980)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Mouse)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517079(CHEMBL4441585)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at mouse CB1R expressed in CHO-K1 cells assessed as CP55940-induced beta-arrestin2 recruitment by pathhunter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of North Carolina At Greensboro

Curated by ChEMBL
LigandPNGBDBM50517079(CHEMBL4441585)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulatory activity at human CB1R expressed in CHO-K1 cells assessed as CP55940-induced cAMP level by hit-hunter cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed