Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50009125
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant H3 receptor expressed in HEK293 cells incubated for 90 minMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Inhibition of rat brain MAO-B using [14C]-phenylethylamine as substrate preincubated for 60 mins followed by substrate addition and measured after 20...More data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant H3 receptor expressed in HEK293 cells incubated for 90 minMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant H3 receptor expressed in HEK293 cells incubated for 90 minMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant H3 receptor expressed in HEK293 cells incubated for 90 minMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 256nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate preincubated for 60 mins followed by substrate addition by discontinuous fluorime...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 991nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate by discontinuous fluorimetric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate preincubated for 30 mins followed by substrate addition by discontinuous fluorime...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 7.92E+3nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate by discontinuous fluorimetric analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H] pyrilamine from human H1 histamine receptorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate preincubated for 60 mins followed by substrate addition by discontinuous fluorime...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H] spiperone from human D3 dopamine receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H] spiperone from human D2 dopamine receptorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate preincubated for 60 mins followed by substrate addition by discontinuous fluorime...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate preincubated for 60 mins followed by substrate addition by discontinuous fluorime...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate by discontinuous fluorimetric analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H] histamine from human H4 histamine receptorMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate by discontinuous fluorimetric analysisMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Human)
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate preincubated for 30 mins followed by substrate addition by discontinuous fluorime...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat brain MAO-B using [14C]-phenylethylamine as substrate preincubated for 60 mins followed by substrate addition and measured after 20...More data for this Ligand-Target Pair
