Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50009477
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataIC50: 48nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529215(CHEMBL342375 | CHEBI:35046)
Affinity DataIC50: 55nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataIC50: 160nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataIC50: 200nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529217(CHEMBL4447214)
Affinity DataIC50: 540nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529216(CHEMBL4444584)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529218(CHEMBL4473641)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Kv7.2 in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
Target1,3-beta-glucan synthase component GSC2(Baker's yeast)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
Target1,3-beta-glucan synthase component GSC2(Baker's yeast)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
Target1,3-beta-glucan synthase component GSC2(Baker's yeast)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
Target1,3-beta-glucan synthase component GSC2(Baker's yeast)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529215(CHEMBL342375 | CHEBI:35046)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of ERG in human HEK293 cells incubated for 1 hr by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of alpha1A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetProtein polybromo-1(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529212(CHEMBL4471453)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of PBR receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529214(CHEMBL343822)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Human)
Marquette University

Curated by ChEMBL
LigandPNGBDBM50529213(CHEMBL4465132)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed