Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50006925
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50504738(CHEMBL4463715)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of recombinant human GABA receptor alpha1beta2gamma2 expressed in CHO cells at 30 uM in presence of GABA and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50504737(CHEMBL4539102)
Affinity DataEC50:  240nMAssay Description:Positive allosteric modulation of recombinant human GABA receptor alpha1beta2gamma2 expressed in CHO cells at 30 uM in presence of GABA and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50504738(CHEMBL4463715)
Affinity DataEC50:  3.08E+3nMAssay Description:Activation of recombinant human GABA receptor alpha1beta2gamma2 expressed in CHO cells in presence of GABA and measured for 120 secs by FMP dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Human)
Qingdao University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50504737(CHEMBL4539102)
Affinity DataEC50:  1.20E+4nMAssay Description:Activation of recombinant human GABA receptor alpha1beta2gamma2 expressed in CHO cells in presence of GABA and measured for 120 secs by FMP dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed