Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50007940
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514172(CHEMBL4536072)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514166(CHEMBL4448448)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514173(CHEMBL4463191)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514167(CHEMBL4560077)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50435396(CHEMBL2391916)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514173(CHEMBL4463191)
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant rat MGL C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514170(CHEMBL4515209)
Affinity DataIC50: 54nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514173(CHEMBL4463191)
Affinity DataIC50: 54nMAssay Description:Inhibition of recombinant rat MGL C201A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514182(CHEMBL3219170)
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50359050(CHEMBL1922513)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM61908(KUC103657N | cid_351236 | 2-methyl-1,2-benzothiazo...)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50435396(CHEMBL2391916)
Affinity DataIC50: 73nMAssay Description:Inhibition of recombinant rat MGL C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514166(CHEMBL4448448)
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant rat MGL C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514180(CHEMBL4439900)
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514166(CHEMBL4448448)
Affinity DataIC50: 114nMAssay Description:Inhibition of recombinant rat MGL C201A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514179(CHEMBL4558017)
Affinity DataIC50: 135nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514183(CHEMBL4445264)
Affinity DataIC50: 163nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514174(CHEMBL4514686)
Affinity DataIC50: 189nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514171(CHEMBL4450432)
Affinity DataIC50: 195nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514172(CHEMBL4536072)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant rat MGL C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514172(CHEMBL4536072)
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant rat MGL C201A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514178(CHEMBL4544505)
Affinity DataIC50: 238nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50435396(CHEMBL2391916)
Affinity DataIC50: 243nMAssay Description:Inhibition of recombinant rat MGL C201A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514176(CHEMBL4449771)
Affinity DataIC50: 278nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM46658(MLS-0254244.0001 | cid_17520 | 1,2-benzothiazol-3-...)
Affinity DataIC50: 307nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514175(CHEMBL4553365)
Affinity DataIC50: 322nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514177(CHEMBL4530292)
Affinity DataIC50: 512nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514181(CHEMBL4438540)
Affinity DataIC50: 568nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50435396(CHEMBL2391916)
Affinity DataIC50: 605nMAssay Description:Inhibition of recombinant rat MGL C201A/C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514169(CHEMBL4576162)
Affinity DataIC50: 759nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514173(CHEMBL4463191)
Affinity DataIC50: 782nMAssay Description:Inhibition of recombinant rat MGL C201A/C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514172(CHEMBL4536072)
Affinity DataIC50: 1.46E+3nMAssay Description:Inhibition of recombinant rat MGL C201A/C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514166(CHEMBL4448448)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of recombinant rat MGL C201A/C208A mutant expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514184(CHEMBL4548018)
Affinity DataIC50: 2.55E+3nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoacylglycerol lipase ABHD6(Mouse)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50435396(CHEMBL2391916)
Affinity DataIC50: 3.58E+3nMAssay Description:Inhibition of mouse ABHD6 expressed in HEK293 cells using 2-AG as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50435396(CHEMBL2391916)
Affinity DataIC50: 9.38E+3nMAssay Description:Inhibition of FAAH in rat brain homogenates using [3H]anandamide as substrate measured after 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetMonoglyceride lipase(Rat)
University of Parma

Curated by ChEMBL
LigandPNGBDBM50514168(CHEMBL4545305)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of recombinant rat MGL expressed in human HeLa cells using 2-oleoylglycerol as substrate preincubated for 10 mins followed by substrate ad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed