Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50006937
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of aromatase in human MCF-7aro cells using [1beta-3H] androstenedione as substrate incubated for 1 hr by liquid scintillation counting met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50504788(CHEMBL4537791)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluorime...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50504787(CHEMBL1371590)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluorime...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50504786(CHEMBL4516755)
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluorime...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed
TargetAromatase(Human)
"G. D'Annunzio" University

Curated by ChEMBL
LigandPNGBDBM50504789(CHEMBL4464506)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human aromatase preincubated for 10 mins followed by substrate and beta-NADP+ addition and measured for 60 mins by fluorime...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/18/2021
Entry Details Article
PubMed