Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50012637
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 250nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM13066({2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid |...)
Affinity DataIC50: 480nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50000541(Leutrol | CHEMBL93 | N-(1-Benzo(b)thien-2-ylethyl)...)
Affinity DataIC50: 630nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558938(CHEMBL4797337)
Affinity DataIC50: 810nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558934(CHEMBL4754218)
Affinity DataIC50: 860nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558934(CHEMBL4754218)
Affinity DataIC50: 980nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558936(CHEMBL4794507)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558937(CHEMBL4779865)
Affinity DataIC50: 4.23E+3nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558936(CHEMBL4794507)
Affinity DataIC50: 4.74E+3nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558937(CHEMBL4779865)
Affinity DataIC50: 5.29E+3nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558935(CHEMBL4742170)
Affinity DataIC50: 6.29E+3nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558938(CHEMBL4797337)
Affinity DataIC50: 8.94E+3nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM13066({2-[(2,6-dichlorophenyl)amino]phenyl}acetic acid |...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558935(CHEMBL4742170)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558941(CHEMBL4779734)
Affinity DataIC50: 1.62E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558944(CHEMBL4764720)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558949(CHEMBL4746020)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558941(CHEMBL4779734)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558942(CHEMBL4757410)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558942(CHEMBL4757410)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558946(CHEMBL4792260)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558945(CHEMBL4776872)
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558943(CHEMBL4777181)
Affinity DataIC50: 3.03E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558934(CHEMBL4754218)
Affinity DataIC50: 3.09E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558940(CHEMBL4750799)
Affinity DataIC50: 3.33E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558949(CHEMBL4746020)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558936(CHEMBL4794507)
Affinity DataIC50: 3.92E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558939(CHEMBL4756619)
Affinity DataIC50: 3.93E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558944(CHEMBL4764720)
Affinity DataIC50: 3.95E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558942(CHEMBL4757410)
Affinity DataIC50: 4.34E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558938(CHEMBL4797337)
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558950(CHEMBL4742772)
Affinity DataIC50: 4.51E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558937(CHEMBL4779865)
Affinity DataIC50: 4.87E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558945(CHEMBL4776872)
Affinity DataIC50: 4.89E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558941(CHEMBL4779734)
Affinity DataIC50: 4.91E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558943(CHEMBL4777181)
Affinity DataIC50: 5.14E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558946(CHEMBL4792260)
Affinity DataIC50: 5.15E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558947(CHEMBL4800127)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558939(CHEMBL4756619)
Affinity DataIC50: 5.35E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558939(CHEMBL4756619)
Affinity DataIC50: 5.35E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558946(CHEMBL4792260)
Affinity DataIC50: 5.62E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558947(CHEMBL4800127)
Affinity DataIC50: 5.65E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558945(CHEMBL4776872)
Affinity DataIC50: 5.66E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558940(CHEMBL4750799)
Affinity DataIC50: 6.24E+4nMAssay Description:Inhibition of recombinant human 5LOX expressed in baculovirus infected Sf insect cells using linoleic acid as substrate preincubated for 5 mins follo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558949(CHEMBL4746020)
Affinity DataIC50: 6.26E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCytochrome c oxidase subunit 2(Human)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558940(CHEMBL4750799)
Affinity DataIC50: 6.39E+4nMAssay Description:Inhibition of recombinant human COX2 expressed in baculovirus infected Sf21 cells using arachidonic acid as substrate preincubated for 5 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558950(CHEMBL4742772)
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Sheep)
University of Malakand

Curated by ChEMBL
LigandPNGBDBM50558944(CHEMBL4764720)
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of sheep COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 5 mins by UV-v...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
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