Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50010430
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
Shoolini University of Biotechnology and Management Sciences

Curated by ChEMBL
LigandPNGBDBM50538770(CHEMBL4637201)
Affinity DataIC50: 8.56E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-3 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
Shoolini University of Biotechnology and Management Sciences

Curated by ChEMBL
LigandPNGBDBM50538769(CHEMBL4646055)
Affinity DataIC50: 9.98E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-3 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Shoolini University of Biotechnology and Management Sciences

Curated by ChEMBL
LigandPNGBDBM50538770(CHEMBL4637201)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Shoolini University of Biotechnology and Management Sciences

Curated by ChEMBL
LigandPNGBDBM50538769(CHEMBL4646055)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in bacterial expression system using ZFR-AMC as substrate measured for 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed