Compile Data Set for Download or QSAR
Report error Found 78 Enz. Inhib. hit(s) with all data for entry = 50007088
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506203(CHEMBL4452312)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506156(CHEMBL4471140)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506173(CHEMBL4589444)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506179(CHEMBL4579583)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506184(CHEMBL4447043)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506187(CHEMBL4522504)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506180(CHEMBL4556573)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506201(CHEMBL4516176)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506178(CHEMBL4555657)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506183(CHEMBL4521017)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506172(CHEMBL4563994)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506185(CHEMBL4438327)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506191(CHEMBL4439570)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506169(CHEMBL4535761)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506162(CHEMBL4463320)
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506157(CHEMBL4517831)
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506198(CHEMBL4539658)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506166(CHEMBL4474747)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506204(CHEMBL4443234)
Affinity DataIC50: 52nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM393615(US09969700, 173)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506195(CHEMBL4438981)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506163(CHEMBL4561582)
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506154(CHEMBL4516450)
Affinity DataIC50: 76nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506177(CHEMBL4452251)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506175(CHEMBL4519162)
Affinity DataIC50: 88nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506186(CHEMBL4449416)
Affinity DataIC50: 92nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506164(CHEMBL4579675)
Affinity DataIC50: 93nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506160(CHEMBL4513970)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human P2X4 receptor expressed in HEK cells assessed as reduction in ATP induced calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 108nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506205(CHEMBL4469574)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Mouse)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 112nMAssay Description:Antagonist activity at mouse P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506182(CHEMBL4593104)
Affinity DataIC50: 134nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506174(CHEMBL4442297)
Affinity DataIC50: 139nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506188(CHEMBL4451946)
Affinity DataIC50: 163nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506200(CHEMBL4443857)
Affinity DataIC50: 173nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506171(CHEMBL4462109)
Affinity DataIC50: 185nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506197(CHEMBL4541425)
Affinity DataIC50: 193nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 211nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Rat)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 233nMAssay Description:Antagonist activity at rat P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of Mg-ATP-induced calcium influx incubated for 30 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506155(CHEMBL4577125)
Affinity DataIC50: 242nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506199(CHEMBL4450002)
Affinity DataIC50: 258nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506194(CHEMBL4462656)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506202(CHEMBL4450779)
Affinity DataIC50: 269nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506206(CHEMBL4451276)
Affinity DataIC50: 317nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506158(CHEMBL4521594)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of inhibition of ATP-evoked current at -90 mV hold...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506153(CHEMBL4444721)
Affinity DataIC50: 345nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506167(CHEMBL4539332)
Affinity DataIC50: 376nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506161(CHEMBL4464823)
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in human 1321N1 cells assessed as inhibition of ATP-induced calcium influx incubated for 15 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetP2X purinoceptor 4(Human)
Bayer

Curated by ChEMBL
LigandPNGBDBM50506168(CHEMBL4533763)
Affinity DataIC50: 441nMAssay Description:Antagonist activity at human P2X4 receptor tranfected in HEK293 cells assessed as inhibition of Bz-ATP-induced calcium influx incubated for 30 mins a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
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