Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50010358
TargetCytochrome P450 1A2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50537942(CHEMBL4645163)
Affinity DataIC50: 960nMAssay Description:Inhibition of recombinant human CYP1A2 using luciferin-ME as substrate preincubated for 10 mins followed by NADPH addition and measured after 10 to 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50537941(CHEMBL4644033)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant human CYP1A2 using luciferin-ME as substrate preincubated for 10 mins followed by NADPH addition and measured after 10 to 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50537940(CHEMBL4640885)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human CYP1A2 using luciferin-ME as substrate preincubated for 10 mins followed by NADPH addition and measured after 10 to 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed