Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50008533
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM247270(US9447029, 2-[2-(3-Pentyloxyphenyl)-ethylamino]-N,...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50520206(CHEMBL4291394)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM161090(US9447029, 2-[2-(3-Butoxyphenyl)-ethylamino]-N,N-d...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50520207(CHEMBL4555166)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50520205(CHEMBL4575754)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Southampton

Curated by ChEMBL
LigandPNGBDBM50520208(CHEMBL4463136)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human ERG assessed as reduction in channel tail current by plate-based planar patch clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed