Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50010503
TargetBifunctional epoxide hydrolase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50264106(CHEMBL3818875)
Affinity DataIC50: 0.0270nMAssay Description:Inhibition of recombinant human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50264106(CHEMBL3818875)
Affinity DataIC50: 0.660nMAssay Description:Inhibition of recombinant human soluble epoxide hydrolase expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50264106(CHEMBL3818875)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50539700(CHEMBL4637413)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50264106(CHEMBL3818875)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of soluble epoxide hydrolase in human whole bloodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50539699(CHEMBL4641357)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM371865(2-[4-Oxo-1-phenyl-8-(1H-pyrazolo[3,4-b]pyridine-5-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant GST-tagged human DDR1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM438155(US10618897, Example 23)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant GST-tagged human DDR1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein-arginine deiminase type-4(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50532282(CHEMBL4539512)
Affinity DataIC50: 50nMAssay Description:Inhibition of PAD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50532282(CHEMBL4539512)
Affinity DataIC50: 250nMAssay Description:Inhibition of PAD4 (unknown origin) in presence of 2 mM CaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM371924(2-[8-(1H-Indazole-5-carbonyl)-4-oxo-1-phenyl-1,3,8...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant GST-tagged human DDR1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM438155(US10618897, Example 23)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant GST-tagged human DDR2 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM371865(2-[4-Oxo-1-phenyl-8-(1H-pyrazolo[3,4-b]pyridine-5-...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of recombinant GST-tagged human DDR2 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM371924(2-[8-(1H-Indazole-5-carbonyl)-4-oxo-1-phenyl-1,3,8...)
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition of recombinant GST-tagged human DDR2 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed