Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50010712
LigandPNGBDBM50541411(CHEMBL4643006)
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of human CLR/RAMP1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50184069(CHEMBL207197 | N-((R)-1-((S)-6-amino-1-oxo-1-(4-(p...)
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541409(CHEMBL4647045)
Affinity DataIC50: 0.0450nMAssay Description:Inhibition of human CLR/RAMP1 by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541412(CHEMBL4644508)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541404(CHEMBL4639133)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50047356(CHEMBL3334624)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541403(CHEMBL4641806)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50047357(CHEMBL3334623)
Affinity DataIC50: 44nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541402(CHEMBL4645875)
Affinity DataIC50: 250nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541401(CHEMBL4634626)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50173483((S)-6-Amino-2-[(R)-3-(3,5-dibromo-4-hydroxy-phenyl...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541408(CHEMBL4643140)
Affinity DataKi:  0.00400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541406(CHEMBL4649325)
Affinity DataKi:  0.00700nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM362044(US9833448, Example 4 | US10272077, Example 4)
Affinity DataKi:  0.0150nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541407(CHEMBL4638635)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM391726(US10300056, Example 11 | N-[(2R)-3-(7-methyl-1H- |...)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM361594(US9833448, Example 1 | US10272077, Example 1)
Affinity DataKi:  0.0670nMAssay Description:Antagonist activity at human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541405(CHEMBL4633407)
Affinity DataKi:  0.110nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541410(CHEMBL4637301)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541413(CHEMBL4649671)
Affinity DataKi:  0.25nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50224431(N-[(3R,6S)-6-(2,3-difluorophenyl)-2-oxo-1-(2,2,2-t...)
Affinity DataKi:  0.770nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
LigandPNGBDBM50541400(CHEMBL4634646)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of human CLR/RAMP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed