Report error Found 409 Enz. Inhib. hit(s) with all data for entry = 50018466
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human USP7 using Ub-Rho110 as substrate by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human USP7 using Ub-Rho110 as substrate by fluorescence based SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human USP7 using Ub-Rho110 as substrate by fluorescence based SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of human USP7 using Ub-Rho as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of human USP7 by SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of human full length his tagged USP7 (208 to 560 residues) expressed in insect sf9 cells using monoubiquitinated ubiquitin-rhodamine as su...More data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Inhibition of human his tagged USP7 (208 to 560 residues) catalytic domain expressed in insect sf9 cells using monoubiquitinated ubiquitin-rhodamine ...More data for this Ligand-Target Pair
Affinity DataEC50: 75nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Inhibition of human USP8 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of human USP7 using ubiquitin-Rh110 as substrate incubated for 30 mins by Fluorometric plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 133nMAssay Description:Inhibition of human USP8 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human USP7 using ubiquitin-Rh110 as substrate incubated for 23 to 45 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 200nMAssay Description:Inhibition of human USP47 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human USP7 using ubiquitin-Rh110 as substrate incubated for 23 to 45 mins by fluorescence based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of human USP8 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of USP8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of USP8 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of human USP8 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human USP7 using Ub-Rho110 as substrate by fluorescence based SPR analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibition of human USP8 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of human USP7 using ubiquitin-Rh110 as substrate incubated for 30 mins by Fluorometric plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of USP47 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of human USP7 using ubiquitin-Rh110 as substrate incubated for 30 mins by Fluorometric plate reader analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Inhibition of human USP47 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataEC50: 360nMAssay Description:Inhibition of human USP47 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 390nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of USP47 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 420nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of human USP7 using Ub-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Inhibition of human recombinant USP7 expressed in Escherichia coli sf9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 424nMAssay Description:Inhibition of human USP7More data for this Ligand-Target Pair
Affinity DataEC50: 430nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Inhibition of USP7 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 450nMAssay Description:Inhibition of human USP47 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataEC50: 470nMAssay Description:Inhibition of human USP7 using Ub-EKL as substrate by SDS-PAGE assayMore data for this Ligand-Target Pair
Affinity DataIC50: 470nMAssay Description:Inhibition of human USP7 using ubiquitin-Rh110 as substrate incubated for 30 mins by Fluorometric plate reader analysisMore data for this Ligand-Target Pair







3D Structure (crystal)




























