Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50007649
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
3D Structure (crystal)TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 27nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 37nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 56nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 93nMAssay Description:Binding affinity to PPARalpha in human MIO-M1 cells assessed as increase in thermal stability preincubated for 3 hrs followed by exposure to 45.5 deg...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 140nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 170nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Binding affinity to PPARalpha in human MIO-M1 cells assessed as increase in thermal stability preincubated for 3 hrs followed by exposure to 45.5 deg...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 540nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 740nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 770nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 810nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 830nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 900nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 960nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 970nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.12E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.18E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 1.61E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 4.43E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 5.32E+3nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 8.52E+3nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataKd: 1.69E+4nMAssay Description:Binding affinity to His-tagged PPARalpha LBD (unknown origin) expressed in Escherichia coli Rosetta (DE3) at 25 degree C by isothermal titration calo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.53E+4nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: 2.56E+4nMAssay Description:Agonist activity at human PPARalpha expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Oklahoma
Curated by ChEMBL
University of Oklahoma
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in nonhuman mammalian cells assessed as increase in receptor transcriptional activity incubated for 22 ...More data for this Ligand-Target Pair
