Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50010934
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50205450((S)-7-(3-(aminomethyl)pyrrolidin-1-yl)-1-cycloprop...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543559(CHEMBL4648309)
Affinity DataIC50: 950nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543557(CHEMBL4636070)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543560(CHEMBL4644781)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543563(CHEMBL4645741)
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543558(CHEMBL4649758)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543561(CHEMBL4642955)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543562(CHEMBL4636102)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543564(CHEMBL4644915)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543565(CHEMBL4638646)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetDNA gyrase A/A/B/B tetramer(Escherichia coli (strain K12))
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50543566(CHEMBL4639662)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase assessed as supercoiling activity by fluorescence assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed