Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50008571
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520569(CHEMBL4456119)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520563(CHEMBL4537710)
Affinity DataIC50: 0.370nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520566(CHEMBL4458123)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520567(CHEMBL4462704)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520562(CHEMBL4533684)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520565(CHEMBL4469271)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520568(CHEMBL4472956)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Usona Institute

Curated by ChEMBL
LigandPNGBDBM50520564(CHEMBL4466148)
Affinity DataIC50: 0.820nMAssay Description:Inhibition of ERalpha in human T47D cells by ERE-driven luciferase reporter gene assay based target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed