Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50013318
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564716(CHEMBL4790926)
Affinity DataIC50: 8nMAssay Description:Inhibition of human CDK9/cyclin T in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564717(CHEMBL4787876)
Affinity DataIC50: 9nMAssay Description:Inhibition of human CDK9/cyclin T in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human CDK9/cyclin T in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564718(CHEMBL4781618)
Affinity DataIC50: 14nMAssay Description:Inhibition of human CDK9/cyclin T in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564719(CHEMBL4793858)
Affinity DataIC50: 15nMAssay Description:Inhibition of human CDK9/cyclin T in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 20nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564720(CHEMBL4788045)
Affinity DataIC50: 59nMAssay Description:Inhibition of human GSK3beta in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564720(CHEMBL4788045)
Affinity DataIC50: 64nMAssay Description:Inhibition of human CDK9/cyclin T in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564720(CHEMBL4788045)
Affinity DataIC50: 70nMAssay Description:Inhibition of human GSK3alpha by ADP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564716(CHEMBL4790926)
Affinity DataIC50: 117nMAssay Description:Inhibition of human GSK3beta in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564716(CHEMBL4790926)
Affinity DataIC50: 121nMAssay Description:Inhibition of human CDK5/p25 in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564718(CHEMBL4781618)
Affinity DataIC50: 160nMAssay Description:Inhibition of human GSK3beta in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564716(CHEMBL4790926)
Affinity DataIC50: 162nMAssay Description:Inhibition of human CDK2/cyclin A in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564717(CHEMBL4787876)
Affinity DataIC50: 195nMAssay Description:Inhibition of human CDK5/p25 in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564719(CHEMBL4793858)
Affinity DataIC50: 216nMAssay Description:Inhibition of human GSK3beta in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 272nMAssay Description:Inhibition of human CDK5/p25 in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564718(CHEMBL4781618)
Affinity DataIC50: 284nMAssay Description:Inhibition of human CDK5/p25 in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564718(CHEMBL4781618)
Affinity DataIC50: 349nMAssay Description:Inhibition of human CDK2/cyclin A in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564717(CHEMBL4787876)
Affinity DataIC50: 356nMAssay Description:Inhibition of human GSK3beta in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 379nMAssay Description:Inhibition of human CDK2/cyclin A in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564717(CHEMBL4787876)
Affinity DataIC50: 469nMAssay Description:Inhibition of human CDK2/cyclin A in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564719(CHEMBL4793858)
Affinity DataIC50: 550nMAssay Description:Inhibition of human CDK5/p25 in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5 activator 1(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564720(CHEMBL4788045)
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human CDK5/p25 in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human GSK3beta in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564719(CHEMBL4793858)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of human CDK2/cyclin A in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
University Paris-Saclay

Curated by ChEMBL
LigandPNGBDBM50564720(CHEMBL4788045)
Affinity DataIC50: 1.73E+3nMAssay Description:Inhibition of human CDK2/cyclin A in presence of ATP by ADP-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed