Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50010619
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540629(CHEMBL4639381)
Affinity DataIC50: 98nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540634(CHEMBL4636738)
Affinity DataIC50: 183nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50006933(CHEMBL3134422)
Affinity DataIC50: 200nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540631(CHEMBL4634711)
Affinity DataIC50: 254nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50109398(CHEMBL2381968)
Affinity DataIC50: 792nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540622(CHEMBL4638389)
Affinity DataIC50: 862nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540633(CHEMBL4645065)
Affinity DataIC50: 1.28E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540621(CHEMBL4645109)
Affinity DataIC50: 1.56E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540635(CHEMBL4642536)
Affinity DataIC50: 1.98E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540618(CHEMBL4648717)
Affinity DataIC50: 2.55E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540628(CHEMBL4642135)
Affinity DataIC50: 2.70E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540619(CHEMBL4649380)
Affinity DataIC50: 3.10E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540630(CHEMBL4639835)
Affinity DataIC50: 4.68E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540632(CHEMBL4635272)
Affinity DataIC50: 5.46E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540620(CHEMBL4641843)
Affinity DataIC50: 5.54E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540624(CHEMBL4647979)
Affinity DataIC50: 5.90E+3nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540626(CHEMBL4633579)
Affinity DataIC50: 2.90E+4nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540623(CHEMBL4648472)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540627(CHEMBL4637259)
Affinity DataIC50: 6.40E+4nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540625(CHEMBL4638535)
Affinity DataIC50: 6.40E+4nMAssay Description:Displacement of AF647-9-mer ETGE peptide from recombinant human biotinylated KEAP1 Kelch domain (322 to 609 residues) expressed in Escherichia coli B...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed