Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50010628
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540727(CHEMBL4642126)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540720(CHEMBL4647613)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540719(CHEMBL4643368)
Affinity DataEC50:  570nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540721(CHEMBL4646200)
Affinity DataEC50:  660nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540725(CHEMBL4637054)
Affinity DataEC50:  780nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540722(CHEMBL4648823)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540724(CHEMBL4646264)
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540717(CHEMBL4643260)
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540723(CHEMBL4638053)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540726(CHEMBL4635505)
Affinity DataEC50:  4.58E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540718(CHEMBL4635684)
Affinity DataEC50:  6.90E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
University of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540728(CHEMBL4644760)
Affinity DataEC50:  9.33E+3nMAssay Description:Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed