Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50010994
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM50543971(CHEMBL4637063)
Affinity DataEC50:  4nMAssay Description:Agonist activity at GAL4-DBD fused human PPARdelta (147 to 441 residues) expressed in HEK293T cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM50543972(CHEMBL4643562)
Affinity DataEC50:  19nMAssay Description:Agonist activity at GAL4-DBD fused human PPARdelta (147 to 441 residues) expressed in HEK293T cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM323618(US10188627, Comparator Cmpd. 2)
Affinity DataEC50:  20nMAssay Description:Agonist activity at N-terminal His-tagged human PPARdelta-LBD expressed in Escherichia coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM50543973(CHEMBL4642511)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at human PPARdelta after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM50543971(CHEMBL4637063)
Affinity DataEC50:  4nMAssay Description:Agonist activity at PPARdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at PPARdelta (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM323618(US10188627, Comparator Cmpd. 2)
Affinity DataEC50:  20nMAssay Description:Transactivation of N-terminal His-tagged human PPARdelta-LBD expressed in Escherichia coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
Daegu-Gyeongbuk Medical Innovation Foundation

Curated by ChEMBL
LigandPNGBDBM50160401(CHEMBL3787648)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed