Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50012866
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataIC50: 369nMAssay Description:Inhibition of human ERG by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataIC50: 2.98E+3nMAssay Description:Inhibition of human ERG by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataKi:  7.80nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataKi:  13nMAssay Description:Binding affinity to 5HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561101(CHEMBL4792709)
Affinity DataKi:  13nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataKi:  16nMAssay Description:Binding affinity to alpha2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561095(CHEMBL4764692)
Affinity DataKi:  16nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561101(CHEMBL4792709)
Affinity DataKi:  21nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561101(CHEMBL4792709)
Affinity DataKi:  21nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  22nMAssay Description:Binding affinity to alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  28nMAssay Description:Binding affinity to alpha2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  39nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561098(CHEMBL4790699)
Affinity DataKi:  42nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  49nMAssay Description:Binding affinity to H1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  54nMAssay Description:Binding affinity to H1 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561094(CHEMBL4777055)
Affinity DataKi:  70nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561105(CHEMBL4799934)
Affinity DataKi:  72nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561096(CHEMBL4755062)
Affinity DataKi:  76nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561094(CHEMBL4777055)
Affinity DataKi:  79nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561095(CHEMBL4764692)
Affinity DataKi:  109nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561094(CHEMBL4777055)
Affinity DataKi:  117nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561105(CHEMBL4799934)
Affinity DataKi:  119nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561098(CHEMBL4790699)
Affinity DataKi:  122nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561099(CHEMBL4760689)
Affinity DataKi:  135nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561100(CHEMBL4764639)
Affinity DataKi:  141nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561098(CHEMBL4790699)
Affinity DataKi:  148nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561099(CHEMBL4760689)
Affinity DataKi:  150nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561105(CHEMBL4799934)
Affinity DataKi:  156nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561090(CHEMBL4779364)
Affinity DataKi:  167nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  186nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  193nMAssay Description:Binding affinity to alpha2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  195nMAssay Description:Binding affinity to alpha1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  224nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561095(CHEMBL4764692)
Affinity DataKi:  258nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  271nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561090(CHEMBL4779364)
Affinity DataKi:  289nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561091(CHEMBL4752919)
Affinity DataKi:  448nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561092(CHEMBL4789422)
Affinity DataKi:  467nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM152525(N-(4-(3-(4-(pyrimidin-2-yl)piperazin-1-yl)propoxy)...)
Affinity DataKi:  498nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  765nMAssay Description:Binding affinity to 5HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  1.14E+3nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  1.19E+3nMAssay Description:Binding affinity to 5HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561102(CHEMBL4794963)
Affinity DataKi:  1.23E+3nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561100(CHEMBL4764639)
Affinity DataKi:  1.59E+3nMAssay Description:Binding affinity to D2 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM50561093(CHEMBL4784373)
Affinity DataKi:  1.99E+3nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Jiangsu Ocean University

Curated by ChEMBL
LigandPNGBDBM152524(N-(4-(3-(4-(pyridin-2-yl)piperazin-1-yl)propoxy)ph...)
Affinity DataKi:  1.99E+3nMAssay Description:Binding affinity to 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
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