Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50018346
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481594(CHEMBL5268220)
Affinity DataKd:  2.11E+4nMAssay Description:Binding affinity to HSP90 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481602(CHEMBL5277647)
Affinity DataKd:  1.00E+3nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481595(CHEMBL5287183)
Affinity DataKd:  36nMAssay Description:Binding affinity to APC (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481596(CHEMBL5277870)
Affinity DataKd: >1.00E+5nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481597(CHEMBL5281856)
Affinity DataKd: >1.50E+4nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481598(CHEMBL5272698)
Affinity DataKd:  8.30E+3nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481599(CHEMBL5283185)
Affinity DataKd:  7.30E+3nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481600(CHEMBL5283334)
Affinity DataKd:  6.00E+3nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481601(CHEMBL5274392)
Affinity DataKd:  3.30E+3nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50369190(CHEMBL4163133)
Affinity DataKi:  15nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition constant by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481602(CHEMBL5277647)
Affinity DataKi:  3.00E+3nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481601(CHEMBL5274392)
Affinity DataKi:  2.20E+4nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481600(CHEMBL5283334)
Affinity DataKi:  2.40E+4nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481599(CHEMBL5283185)
Affinity DataKi:  3.20E+4nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481595(CHEMBL5287183)
Affinity DataKi:  4.46E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition constant by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481598(CHEMBL5272698)
Affinity DataKi:  5.80E+4nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481597(CHEMBL5281856)
Affinity DataKi: >5.00E+5nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetHistone-lysine N-methyltransferase 2A(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50481596(CHEMBL5277870)
Affinity DataKi: >1.00E+6nMAssay Description:Competitive binding affinity to full length wild type MLL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed