Report error Found 89 Enz. Inhib. hit(s) with all data for entry = 50012048
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of FITC-diclofenac from human plasma derived TTR measured after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.26E+3nMAssay Description:Displacement of FITC-diclofenac from human plasma derived TTR measured after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of FITC-diclofenac from human plasma derived TTR measured after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 1.67E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+3nMAssay Description:Displacement of FITC-diclofenac from human plasma derived TTR measured after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of FITC-diclofenac from human plasma derived TTR measured after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from MBP-tagged RBP4 (unknown origin) expressed in Escherichia coli assessed as reduction in untagged Eu-label...More data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.35E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 2.44E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.85E+3nMAssay Description:Displacement of FITC-diclofenac from human plasma derived TTR measured after overnight incubation by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetRetinol-binding protein 4(Human)
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Albany College of Pharmacy and Health Sciences
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of [3H]-all-trans-retinol from biotinylated human urine derived RBP4 measured after 16 hrs by scintillation proximity assayMore data for this Ligand-Target Pair





























