Compile Data Set for Download or QSAR
Report error Found 132 Enz. Inhib. hit(s) with all data for entry = 50012061
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553771(CHEMBL4776986)
Affinity DataKi:  0.00300nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553769(CHEMBL4798887)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553767(CHEMBL4789659)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human MOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553779(CHEMBL4742999)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553770(CHEMBL4758754)
Affinity DataKi:  0.160nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553767(CHEMBL4789659)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553768(CHEMBL4744531)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553768(CHEMBL4744531)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553772(CHEMBL4749016)
Affinity DataKi:  0.320nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553775(CHEMBL4745899)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553767(CHEMBL4789659)
Affinity DataKi:  0.430nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553777(CHEMBL4597094)
Affinity DataKi:  0.460nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553776(CHEMBL4747286)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  0.550nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553769(CHEMBL4798887)
Affinity DataKi:  0.780nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553771(CHEMBL4776986)
Affinity DataEC50:  0.860nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553769(CHEMBL4798887)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553767(CHEMBL4789659)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human DOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553769(CHEMBL4798887)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-Diprenorphine from recombinant human delta opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553773(CHEMBL4742666)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553775(CHEMBL4745899)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553777(CHEMBL4597094)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553773(CHEMBL4742666)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553771(CHEMBL4776986)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553772(CHEMBL4749016)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553779(CHEMBL4742999)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553768(CHEMBL4744531)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553778(CHEMBL4740539)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553780(CHEMBL4762684)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS2 stably expressed in human 1321N1 cell membranes incubated for 60 mins by gamma counter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553777(CHEMBL4597094)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553770(CHEMBL4758754)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553771(CHEMBL4776986)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553776(CHEMBL4747286)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553766(CHEMBL4761165)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553773(CHEMBL4742666)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human MOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553768(CHEMBL4744531)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50070386(CHEMBL3408737)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human MOR expressed in human U2OS cells assessed as increase in beta arrestin2 recruitment incubated for 90 mins by pathhunter be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553774(CHEMBL4750783)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553775(CHEMBL4745899)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at human MOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553775(CHEMBL4745899)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at human NTS1 expressed in HEK293 cells co-expressing Galphaq/RlucII/GFP10-Ggamma1/Gbeta1 assessed as increase in Galphaq activation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553772(CHEMBL4749016)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553770(CHEMBL4758754)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]-DAMGO from recombinant human mu opioid receptor expressed in CHO cell membrane incubated for 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553769(CHEMBL4798887)
Affinity DataEC50:  9.10nMAssay Description:Agonist activity at human MOR stably expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by liquid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50553775(CHEMBL4745899)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]-neurotensin from human recombinant NTS1 stably expressed in CHO-K1 cell membranes incubated for 60 mins by gamma counter metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
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