Compile Data Set for Download or QSAR
Report error Found 67 Enz. Inhib. hit(s) with all data for entry = 50018373
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607881(CHEMBL5282218)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human MAO-B using tyramine as substrate by amplex red assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607883(CHEMBL5275814)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of rat brain mitochondria MAO-B using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured for 15 by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607884(CHEMBL5266605)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of rat brain mitochondria MAO-B using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured for 15 by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50606832(CHEMBL5219522)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate incubated for 6 mins followed by substrate addition by DTNB reagent based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607857(CHEMBL5279129)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured upto 20 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50606832(CHEMBL5219522)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured upto 20 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607880(CHEMBL5269376)
Affinity DataIC50: 12nMAssay Description:Inhibition of human MAO-B using tyramine as substrate by amplex red assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50553263(CHEMBL4790416)
Affinity DataIC50: 18nMAssay Description:Inhibition of human MAO-A using p-tyramine as substrate preincubated for 15 mins followed by substrate addition and measured after 30 mins by Ample r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607863(CHEMBL5267475)
Affinity DataIC50: 28nMAssay Description:Inhibition of MAO-B (unknown origin) using tyramine hydrochloride as substrate incubated for 30 mins followed by substrate addition and measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607873(CHEMBL5286562)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human MAO-B expressed in baculovirus-infected BTI insect cells using p-tyramine as substrate incubated for 45 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50553263(CHEMBL4790416)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human AChE using acetylcholine as substrate preincubated for 15 mins followed by substrate addition and measured after 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Mouse)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607871(CHEMBL5280820)
Affinity DataIC50: 32nMAssay Description:Inhibition of mouse AChE using acetylthiocholine iodide as substrate incubated for 20 mins by DTNB reagent based Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607866(CHEMBL227391)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate incubated for 20 min by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607878(CHEMBL5285071)
Affinity DataIC50: 34nMAssay Description:Inhibition of rat brain mitochondria MAO-B using benzylamine as substrate incubated for 30 mins by microplate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607865(CHEMBL5286673)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 10 mins followed by substrate addition and measured 20 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human MAO-B using tyramine hydrochloride as substrate preincubated for 30 mins followed by substrate addition and measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607856(CHEMBL5283994)
Affinity DataIC50: 44nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate incubated for 6 mins followed by substrate addition by DTNB reagent based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607870(CHEMBL5278526)
Affinity DataIC50: 49nMAssay Description:Inhibition of MAO-B (unknown origin) using as tyramine as substrate by Ampliflu red reagent based fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607879(CHEMBL5289674)
Affinity DataIC50: 52nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate incubated for 15 mins by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607869(CHEMBL2238112)
Affinity DataIC50: 54nMAssay Description:Inhibition of MAO-B (unknown origin) using as tyramine as substrate by Ampliflu red reagent based fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607855(CHEMBL5266061)
Affinity DataIC50: 56nMAssay Description:Inhibition of MAO-B (unknown origin) using tyramine hydrochloride as substrate incubated for 30 mins by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607794(CHEMBL1360330)
Affinity DataIC50: 87nMAssay Description:Inhibition of MAO-B (unknown origin) using benzylamine as substrate by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607885(CHEMBL5269911)
Affinity DataIC50: 97nMAssay Description:Inhibition of human MAO-B using tyramine hydrochloride as substrate preincubated for 30 mins followed by substrate addition and measured after 30 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50606833(CHEMBL5219483)
Affinity DataIC50: 101nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured upto 20 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607856(CHEMBL5283994)
Affinity DataIC50: 101nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured upto 20 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50606833(CHEMBL5219483)
Affinity DataIC50: 114nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate incubated for 6 mins followed by substrate addition by DTNB reagent based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607868(CHEMBL2088271)
Affinity DataIC50: 114nMAssay Description:Inhibition of MAO-B (unknown origin) using as tyramine as substrate by Ampliflu red reagent based fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM23413(5-hydroxy-7-methoxy-2-(4-methoxyphenyl)-4H-chromen...)
Affinity DataIC50: 198nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate preincubated for 10 mins followed by substrate addition and measured after 20 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50487758(CHEBI:59979 | Tricin)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 10 mins followed by substrate addition and measured for 20 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607875(CHEMBL5277488)
Affinity DataIC50: 342nMAssay Description:Inhibition of recombinant human MAO-B using tyramine hydrochloride as substrate preincubated for 30 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607864(CHEMBL5279769)
Affinity DataIC50: 372nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate incubated for 20 min by fluorescent spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607867(CHEMBL5283324)
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant human MAO-B expressed in insect cells using kynuramine as substrate incubated for 20 mins by Amplex Red reagent based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607859(CHEMBL293718)
Affinity DataIC50: 444nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 20 mins followed by substrate addition by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607874(CHEMBL5270248)
Affinity DataIC50: 540nMAssay Description:Inhibition of human AChE using acetylcholine as substrate incubated for 5 mins followed by substrate addition by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607858(CHEMBL5289375)
Affinity DataIC50: 560nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 20 mins followed by substrate addition by spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607872(CHEMBL5286976)
Affinity DataIC50: 638nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate incubated for 20 mins by fluorescence spectrophotometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM19459(Prunetol | Genisteol | CHEMBL44 | US8552057, 2 | c...)
Affinity DataIC50: 650nMAssay Description:Inhibition of recombinant human MAO-B using kynuramine as substrate preincubated for 10 mins followed by substrate addition and measured after 20 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCholinesterase(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50553263(CHEMBL4790416)
Affinity DataIC50: 666nMAssay Description:Inhibition of human BuChE using butyrylthiocholine iodide as substrate preincubated for 30 mins followed by substrate addition and measured after 15 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 10 mins followed by substrate addition and measured for 20 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50276157(CHEMBL483526 | Alternariol 5-O-Methyl Ether)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of human MAO-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607865(CHEMBL5286673)
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate incubated for 10 mins followed by substrate addition and measured 20 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607871(CHEMBL5280820)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human MAO-B using benzylamine as substrate preincubated for 15 mins followed by substrate addition and measured after 15 mins by fluore...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50410873(CHEMBL105360 | CHEBI:65737)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of human MAO-B using benzylamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50059989(cid_5324473 | CHEMBL105350 | 1,7-bis(4-hydroxyphen...)
Affinity DataIC50: 2.59E+3nMAssay Description:Inhibition of human MAO-B using benzylamine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAcetylcholinesterase(Electric eel)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50519770(CHEMBL3939546)
Affinity DataIC50: 3.04E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607867(CHEMBL5283324)
Affinity DataIC50: 3.63E+3nMAssay Description:Inhibition of recombinant human MAO-A expressed in insect cells using kynuramine as substrate incubated for 20 mins by Amplex Red reagent based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50110725(CHEMBL18116 | 5-(hydroxymethyl)-3-(3-methylphenyl)...)
Affinity DataIC50: 3.92E+3nMAssay Description:Inhibition of human MAO-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607874(CHEMBL5270248)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of recombinant human MAO-B using p-tyramine as substrate preincubated for 15 mins followed by substrate addition and measured after 20 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607856(CHEMBL5283994)
Affinity DataIC50: 5.85E+3nMAssay Description:Inhibition of recombinant human MAO-A using p-tyramine as substrate incubated for 15 mins followed by substrate addition and measured for 15 to 20 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Jamia Millia Islamia

Curated by ChEMBL
LigandPNGBDBM50607862(CHEMBL5286281)
Affinity DataIC50: 6.12E+3nMAssay Description:Inhibition of recombinant human MAO-A using kynuramine as substrate incubated for 10 mins followed by substrate addition and measured for 20 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
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