Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50012084
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554030(CHEMBL4756339)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554031(CHEMBL4749110)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554033(CHEMBL4794201)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554032(CHEMBL4741135)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50199195(CHEMBL3892042 | US10131658, Compound 8)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554033(CHEMBL4794201)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of alpha5beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of alpha5beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472679(US10836720, HIJ-1017)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472684(US10836720, HIJ-1018)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554032(CHEMBL4741135)
Affinity DataIC50: 1nMAssay Description:Inhibition of alpha5beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554031(CHEMBL4749110)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of alpha5beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554030(CHEMBL4756339)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of alpha5beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472676(US10836720, HIJ-1016)
Affinity DataIC50: 4nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472698(US10836720, HIJ-1437)
Affinity DataIC50: 32nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472689(US10836720, HIJ-1094)
Affinity DataIC50: 32nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472689(US10836720, HIJ-1094)
Affinity DataIC50: 40nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472690(US10836720, HIJ-1099)
Affinity DataIC50: 50nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-4/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554031(CHEMBL4749110)
Affinity DataIC50: 100nMAssay Description:Inhibition of alpha4beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-4/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 105nMAssay Description:Inhibition of alpha4beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554029(CHEMBL4750022)
Affinity DataIC50: 110nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-4/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554030(CHEMBL4756339)
Affinity DataIC50: 136nMAssay Description:Inhibition of alpha4beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472690(US10836720, HIJ-1099)
Affinity DataIC50: 158nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-4/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554032(CHEMBL4741135)
Affinity DataIC50: 161nMAssay Description:Inhibition of alpha4beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-4/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554033(CHEMBL4794201)
Affinity DataIC50: 182nMAssay Description:Inhibition of alpha4beta1 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472686(US10836720, HIJ-1083)
Affinity DataIC50: 316nMAssay Description:Inhibition of alphavbeta1 integrin (unknown origin) expressed in CHO cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554033(CHEMBL4794201)
Affinity DataIC50: 320nMAssay Description:Inhibition of alphavbeta5 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472679(US10836720, HIJ-1017)
Affinity DataIC50: 500nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472686(US10836720, HIJ-1083)
Affinity DataIC50: 830nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472684(US10836720, HIJ-1018)
Affinity DataIC50: 900nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554032(CHEMBL4741135)
Affinity DataIC50: 980nMAssay Description:Inhibition of alphavbeta5 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472689(US10836720, HIJ-1094)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of alphavbeta3 integrin (unknown origin) expressed in human SW480 cells transfected with human beta3 assessed as inhibition of cell adhesi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554033(CHEMBL4794201)
Affinity DataIC50: 1.87E+3nMAssay Description:Inhibition of alphavbeta6 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of alphavbeta6 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of alphavbeta5 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472690(US10836720, HIJ-1099)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of alphavbeta3 integrin (unknown origin) expressed in human SW480 cells transfected with human beta3 assessed as inhibition of cell adhesi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554033(CHEMBL4794201)
Affinity DataIC50: 6.83E+3nMAssay Description:Inhibition of alphavbeta8 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 8.80E+3nMAssay Description:Inhibition of alphavbeta3 integrin (unknown origin) expressed in human SW480 cells transfected with human beta3 assessed as inhibition of cell adhesi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472676(US10836720, HIJ-1016)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554031(CHEMBL4749110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta6 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-5(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554031(CHEMBL4749110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta5 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554032(CHEMBL4741135)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta6 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM472699(US10836720, HIJ-1483)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta8 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554030(CHEMBL4756339)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta8 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554031(CHEMBL4749110)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta8 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554032(CHEMBL4741135)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta8 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50199195(CHEMBL3892042 | US10131658, Compound 8)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alpha5beta1 integrin in human SW480 cells assessed as inhibition of cell adhesion to fibronectin incubated for 60 mins by crystal viole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
University of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50554030(CHEMBL4756339)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of alphavbeta6 integrin (unknown origin) by solid phase binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
Displayed 1 to 50 (of 62 total ) | Next | Last >>
Jump to: