Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50012329
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556595(CHEMBL4740154)
Affinity DataIC50: 0.320nMAssay Description:Antagonist activity at human H3 receptor expressed in HEK293 cells centrifuged for 3 mins followed by 60 mins incubation by LANCE Ultra cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556588(CHEMBL4752838)
Affinity DataIC50: 640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556587(CHEMBL4791397)
Affinity DataIC50: 640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556586(CHEMBL4781670)
Affinity DataIC50: 640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556585(CHEMBL4751314)
Affinity DataIC50: 640nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556593(CHEMBL4751815)
Affinity DataIC50: 680nMAssay Description:Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells using p-Tyramine as substrate incubated for 15 mins by fluorescence meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556590(CHEMBL4778798)
Affinity DataIC50: 860nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556594(CHEMBL4750523)
Affinity DataIC50: 860nMAssay Description:Inhibition of human MAO-B expressed in baculovirus infected BTI insect cells using p-Tyramine as substrate incubated for 15 mins by fluorescence meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556589(CHEMBL4758784)
Affinity DataIC50: 960nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556595(CHEMBL4740154)
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation incubated for 24 hrs by ThT fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556584(CHEMBL4744947)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by ThT fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556583(CHEMBL4755924)
Affinity DataIC50: 7.05E+3nMAssay Description:Inhibition of self-induced amyloid beta (1 to 42) (unknown origin) aggregation by ThT fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556581(CHEMBL4743941)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556582(CHEMBL4797501)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556580(CHEMBL4757329)
Affinity DataIC50: 4.88E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556591(CHEMBL4763495)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50086229(CHEMBL326815)
Affinity DataIC50: 2.10E+5nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcetylcholinesterase(Pacific electric ray)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50556592(CHEMBL4777813)
Affinity DataIC50: 2.46E+5nMAssay Description:Inhibition of Torpedo californica AChE using acetylthiocholine iodide as substrate preincubated for 15 mins followed by substrate addition and measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed