Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50012934
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561646(CHEMBL4798102)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM64682(US9475819, 10A)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50203731(CHEMBL3973097)
Affinity DataKi:  5.20nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50438822(CHEMBL2413367)
Affinity DataKi:  6nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163902(US9475819, 33 | US9062078, 33 | US9695183, 33 | US...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM65032(US9475819, 279)
Affinity DataKi:  9nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163879(US9475819, 11 | US9062078, 11 | US9695183, 12B | U...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163876(US9475819, 9 | US9062078, 9 | US9695183, 10B | US9...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163879(US9475819, 11 | US9062078, 11 | US9695183, 12B | U...)
Affinity DataKi:  13nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM64646(US9475819, 8A)
Affinity DataKi:  14nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561653(CHEMBL4749384)
Affinity DataKi:  14nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561652(CHEMBL4752792)
Affinity DataKi:  15nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561651(CHEMBL4786307)
Affinity DataKi:  16nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM4535(US9475819, 5A)
Affinity DataKi:  18nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM4532(US9475819, 3B)
Affinity DataKi:  19nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561647(CHEMBL4750440)
Affinity DataKi:  19nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561648(CHEMBL4743991)
Affinity DataKi:  25nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM65030(US9475819, 181)
Affinity DataKi:  30nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM64682(US9475819, 10A)
Affinity DataKi:  32nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163902(US9475819, 33 | US9062078, 33 | US9695183, 33 | US...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163901(US9475819, 32 | US9062078, 32 | US9695183, 32 | US...)
Affinity DataKi:  41nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50384416(CHEMBL291536 | CHEMBL2111553 | SB-334867)
Affinity DataKi:  48nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM164066(US9475819, 196 | US9062078, 196 | US9695183, 196 |...)
Affinity DataKi:  52nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163899(US9475819, 30 | US9062078, 30 | US9695183, 30 | US...)
Affinity DataKi:  59nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561650(CHEMBL4747380)
Affinity DataKi:  61nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM164050(US9475819, 182 | US9062078, 181 | US9695183, 183b ...)
Affinity DataKi:  62nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561649(CHEMBL4797068)
Affinity DataKi:  65nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163876(US9475819, 9 | US9062078, 9 | US9695183, 10B | US9...)
Affinity DataKi:  72nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM164057(US9475819, 187 | US9062078, 187 | US9695183, 187 |...)
Affinity DataKi:  75nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM164081(US9475819, 211 | US9062078, 211 | US9695183, 211 |...)
Affinity DataKi:  96nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM326730((R/S)-(3-fluoro-2-(pyrimidin-2-yl)phenyl)(2-((5-(t...)
Affinity DataKi:  100nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM64646(US9475819, 8A)
Affinity DataKi:  110nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM326704((R/S)-(2-(2H-1,2,3-triazol-2-yl)phenyl)-2-((5-(tri...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM326712((R/S)-(3-fluoro-2-(pyrimidin-2-yl)phenyl)-2-((5-(t...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163901(US9475819, 32 | US9062078, 32 | US9695183, 32 | US...)
Affinity DataKi:  160nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM164091(US9475819, 221 | US9062078, 221 | US9695183, 221 |...)
Affinity DataKi:  180nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163899(US9475819, 30 | US9062078, 30 | US9695183, 30 | US...)
Affinity DataKi:  200nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM4532(US9475819, 3B)
Affinity DataKi:  230nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50438822(CHEMBL2413367)
Affinity DataKi:  417nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163916(US9475819, 47 | US9062078, 47 | US9695183, 47 | US...)
Affinity DataKi:  420nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM4535(US9475819, 5A)
Affinity DataKi:  430nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM163916(US9475819, 47 | US9062078, 47 | US9695183, 47 | US...)
Affinity DataKi:  500nMAssay Description:Binding affinity to human OXIRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561647(CHEMBL4750440)
Affinity DataKi:  520nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561653(CHEMBL4749384)
Affinity DataKi:  540nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561648(CHEMBL4743991)
Affinity DataKi:  560nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM164057(US9475819, 187 | US9062078, 187 | US9695183, 187 |...)
Affinity DataKi:  620nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561651(CHEMBL4786307)
Affinity DataKi:  700nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561649(CHEMBL4797068)
Affinity DataKi:  730nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM65030(US9475819, 181)
Affinity DataKi:  770nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50561646(CHEMBL4798102)
Affinity DataKi:  1.01E+3nMAssay Description:Binding affinity to human OX2RMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
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