Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50013684
TargetDual specificity mitogen-activated protein kinase kinase 4(Mouse)
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50396483(PLX-4032 | RG 7204 | Ro 5185426 | VEMURAFENIB | US...)
Affinity DataKd:  8.20nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Mouse)
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50568578(CHEMBL4868537)
Affinity DataKd:  3.5nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Mouse)
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50568579(CHEMBL4848804)
Affinity DataKd:  0.850nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Mouse)
Eberhard Karls Universit£T T£Bingen

Curated by ChEMBL
LigandPNGBDBM50568580(CHEMBL4857316)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed