Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50012948
TargetOrexin receptor type 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50561747(CHEMBL4740509)
Affinity DataIC50: 0.230nMAssay Description:Agonist activity at human recombinant OX2R expressed in CHOK1 cells assessed as increase in intracellular Ca2+ mobilization by measuring IP3 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM514632(US11098029, Example 67)
Affinity DataIC50: 0.230nMAssay Description:Agonist activity at human recombinant OX2R expressed in CHOK1 cells assessed as increase in intracellular Ca2+ mobilization by measuring IP3 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM514589(US11098029, Example 25)
Affinity DataIC50: 0.270nMAssay Description:Agonist activity at human recombinant OX2R expressed in CHOK1 cells assessed as increase in intracellular Ca2+ mobilization by measuring IP3 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM514632(US11098029, Example 67)
Affinity DataIC50: 0.460nMAssay Description:Agonist activity at human recombinant OX2R expressed in CHOK1 cells assessed as increase in intracellular Ca2+ mobilization by measuring IP3 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50561746(CHEMBL4799832)
Affinity DataIC50: 0.470nMAssay Description:Agonist activity at human recombinant OX2R expressed in CHOK1 cells assessed as increase in intracellular Ca2+ mobilization by measuring IP3 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM514582(US11098029, Example 18)
Affinity DataIC50: 0.5nMAssay Description:Agonist activity at human recombinant OX2R expressed in CHOK1 cells assessed as increase in intracellular Ca2+ mobilization by measuring IP3 producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed