Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50012975
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561918(CHEMBL4761849)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561919(CHEMBL4781389)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561920(CHEMBL4764969)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561921(CHEMBL4778498)
Affinity DataEC50:  13nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561922(CHEMBL4799017)
Affinity DataEC50:  16nMAssay Description:Agonist activity at RXFP3 (unknown origin) stably expressed in CHO-K1 cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561918(CHEMBL4761849)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561919(CHEMBL4781389)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561920(CHEMBL4764969)
Affinity DataEC50:  19nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561921(CHEMBL4778498)
Affinity DataEC50:  282nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561922(CHEMBL4799017)
Affinity DataEC50:  14nMAssay Description:Agonist activity at RXFP4 (unknown origin) stably expressed in CHO cells co-transfected with pCRE assessed as inhibition of forskolin-induced cAMP ac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561918(CHEMBL4761849)
Affinity DataKi:  46nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561920(CHEMBL4764969)
Affinity DataKi:  110nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561919(CHEMBL4781389)
Affinity DataKi:  186nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561922(CHEMBL4799017)
Affinity DataKi:  191nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 1(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50561921(CHEMBL4778498)
Affinity DataKi:  331nMAssay Description:Displacement of Eu-labeled H3B1-22R from RXFP3 (unknown origin) stably expressed in CHO-K1 cells by competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed