Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50018389
TargetEpidermal growth factor receptor(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607953(CHEMBL5279539)
Affinity DataIC50: 21nMAssay Description:Inhibition of wild type human EGFR measured by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607954(CHEMBL5266361)
Affinity DataIC50: 56nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607956(CHEMBL3186763)
Affinity DataIC50: 82nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607952(CHEMBL5291481)
Affinity DataIC50: 102nMAssay Description:Inhibition of wild type human EGFR measured by ELISA analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607957(CHEMBL5279820)
Affinity DataIC50: 140nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607954(CHEMBL5266361)
Affinity DataIC50: 420nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607957(CHEMBL5279820)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607955(CHEMBL5281174)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of PI3Kdelta (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607954(CHEMBL5266361)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607957(CHEMBL5279820)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607956(CHEMBL3186763)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607955(CHEMBL5281174)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607956(CHEMBL3186763)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kgamma (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Rat)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607955(CHEMBL5281174)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha in rat Rat1 cells reduction in phosphorylation of AKT at Ser473 residue incubated for 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Rat)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607954(CHEMBL5266361)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha in rat Rat1 cells reduction in phosphorylation of AKT at Ser473 residue incubated for 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Rat)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607957(CHEMBL5279820)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha in rat Rat1 cells reduction in phosphorylation of AKT at Ser473 residue incubated for 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Rat)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607956(CHEMBL3186763)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha in rat Rat1 cells reduction in phosphorylation of AKT at Ser473 residue incubated for 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607955(CHEMBL5281174)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3Kalpha (unknown origin) incubated for 90 mins by [gamma-33P]-ATP based scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetThermolysin(Bacillus thermoproteolyticus)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607951(CHEMBL1164912)
Affinity DataKi:  5.93E+4nMAssay Description:Binding affinity to Bacillus thermoproteolyticus Thermolysin assessed as inhibition constant by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetThermolysin(Bacillus thermoproteolyticus)
Universita Degli Studi di Palermo

Curated by ChEMBL
LigandPNGBDBM50607951(CHEMBL1164912)
Affinity DataIC50: 7.69E+4nMAssay Description:Inhibition of Bacillus thermoproteolyticus ThermolysinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed