Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50013100
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562673(CHEMBL4761606)
Affinity DataEC50:  19nMAssay Description:Agonist activity at CB2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562678(CHEMBL4763456)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562677(CHEMBL4747832)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562676(CHEMBL4742310)
Affinity DataEC50:  676nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562678(CHEMBL4763456)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562677(CHEMBL4747832)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562676(CHEMBL4742310)
Affinity DataEC50:  673nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562675(CHEMBL4763316)
Affinity DataEC50:  6.76E+3nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562674(CHEMBL4760835)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562675(CHEMBL4763316)
Affinity DataEC50:  6.76E+3nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562674(CHEMBL4760835)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human CB2 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human CB1 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human CB1 expressed in mouse AtT20 cells assessed as activation of G-protein gated inwardly rectifying K+ channels measured every...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562673(CHEMBL4761606)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CB1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562673(CHEMBL4761606)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-CP55940 from human CB2 expressed in CHO cell membrane incubated for 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562678(CHEMBL4763456)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-CP55940 from human CB2 expressed in CHO cell membrane incubated for 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562673(CHEMBL4761606)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 expressed in CHO cell membrane incubated for 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562679(CHEMBL4752252)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 expressed in CHO cell membrane incubated for 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562678(CHEMBL4763456)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB1 expressed in CHO cell membrane incubated for 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50562679(CHEMBL4752252)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from human CB2 expressed in CHO cell membrane incubated for 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed