Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50012981
Target5'-nucleotidase(Human)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561931(CHEMBL4746318)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Human)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561933(CHEMBL4788305)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561936(CHEMBL4741833)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Human)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561932(CHEMBL4761451)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Human)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561938(CHEMBL4746633)
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes using AMP as substrate preincubated for 10 mins followed by sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Human)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561930(CHEMBL4760778)
Affinity DataIC50: 460nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561931(CHEMBL4746318)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561934(CHEMBL4753669)
Affinity DataIC50: 680nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Human)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561929(CHEMBL4797703)
Affinity DataIC50: 690nMAssay Description:Inhibition of recombinant human ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561937(CHEMBL4780721)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561935(CHEMBL4761355)
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561933(CHEMBL4788305)
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561932(CHEMBL4761451)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
Target5'-nucleotidase(Rat)
Bahauddin Zakariya University

Curated by ChEMBL
LigandPNGBDBM50561930(CHEMBL4760778)
Affinity DataIC50: 7.99E+3nMAssay Description:Inhibition of recombinant rat ecto-5' nucleotidase expressed in COS7 cell membranes assessed as inorganic phosphate release using AMP as substrate uM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed