Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50011478
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataEC50:  7.90nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547990(CHEMBL4799795)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547991(CHEMBL4740938)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547992(CHEMBL4754473)
Affinity DataEC50:  8.30nMAssay Description:Agonist activity at human RXFP4 transfected in CHO-K1 cells co-transfected with pCRE-beta-galactosidase reporter plasmid assessed as inhibition of fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547989(CHEMBL4747872)
Affinity DataKi:  35nMAssay Description:Competitive binding affinity to human RXFP4 receptor transfected in CHO-K1 cells in presence of europium-labeled Eu(A)-R3/I5 by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547990(CHEMBL4799795)
Affinity DataKi:  35nMAssay Description:Competitive binding affinity to human RXFP4 receptor transfected in CHO-K1 cells in presence of europium-labeled Eu(A)-R3/I5 by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetRelaxin-3 receptor 2(Human)
University of Melbourne

Curated by ChEMBL
LigandPNGBDBM50547991(CHEMBL4740938)
Affinity DataKi:  50nMAssay Description:Competitive binding affinity to human RXFP4 receptor transfected in CHO-K1 cells in presence of europium-labeled Eu(A)-R3/I5 by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed