Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50013444
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565940(CHEMBL4787835)
Affinity DataIC50: 0.240nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565948(CHEMBL4780301)
Affinity DataIC50: 0.260nMAssay Description:Binding affinity to human integrin alphaVbeta6 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565938(CHEMBL4798050)
Affinity DataIC50: 0.340nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565937(CHEMBL4782291)
Affinity DataIC50: 0.350nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565939(CHEMBL4794071)
Affinity DataIC50: 0.430nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565942(CHEMBL4790959)
Affinity DataIC50: 0.520nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565943(CHEMBL4787559)
Affinity DataIC50: 0.520nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565941(CHEMBL4798169)
Affinity DataIC50: 0.530nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565934(CHEMBL4791029)
Affinity DataIC50: 0.530nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 0.540nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565945(CHEMBL4795994)
Affinity DataIC50: 0.590nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565933(CHEMBL4798049)
Affinity DataIC50: 0.620nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565944(CHEMBL4793182)
Affinity DataIC50: 0.740nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565947(CHEMBL4787675)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50004058(N-(butylsulfonyl)-O-(4-piperidin-4-ylbutyl)-L-tyro...)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity to human integrin alpha2bbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565935(CHEMBL4800039)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565946(CHEMBL4787900)
Affinity DataIC50: 5.10nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565947(CHEMBL4787675)
Affinity DataIC50: 9.90nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565935(CHEMBL4800039)
Affinity DataIC50: 10nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50235980(CHEMBL429876 | EMD-121974 | cyclo(Arg-Gly-Asp-D-Ph...)
Affinity DataIC50: 15nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565943(CHEMBL4787559)
Affinity DataIC50: 22nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565948(CHEMBL4780301)
Affinity DataIC50: 24nMAssay Description:Binding affinity to human integrin alphaVbeta8 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565945(CHEMBL4795994)
Affinity DataIC50: 32nMAssay Description:Binding affinity to human integrin alphaVbeta6 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565942(CHEMBL4790959)
Affinity DataIC50: 36nMAssay Description:Binding affinity to human integrin alphaVbeta6 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565943(CHEMBL4787559)
Affinity DataIC50: 39nMAssay Description:Binding affinity to human integrin alphaVbeta8 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565940(CHEMBL4787835)
Affinity DataIC50: 39nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565941(CHEMBL4798169)
Affinity DataIC50: 43nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565939(CHEMBL4794071)
Affinity DataIC50: 49nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565944(CHEMBL4793182)
Affinity DataIC50: 50nMAssay Description:Binding affinity to human integrin alphaVbeta6 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565943(CHEMBL4787559)
Affinity DataIC50: 54nMAssay Description:Binding affinity to human integrin alphaVbeta6 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565937(CHEMBL4782291)
Affinity DataIC50: 58nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565944(CHEMBL4793182)
Affinity DataIC50: 66nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565933(CHEMBL4798049)
Affinity DataIC50: 74nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565944(CHEMBL4793182)
Affinity DataIC50: 77nMAssay Description:Binding affinity to human integrin alphaVbeta8 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565938(CHEMBL4798050)
Affinity DataIC50: 91nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565945(CHEMBL4795994)
Affinity DataIC50: 193nMAssay Description:Binding affinity to human integrin alphaVbeta8 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565942(CHEMBL4790959)
Affinity DataIC50: 220nMAssay Description:Binding affinity to human integrin alphaVbeta8 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-6(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565946(CHEMBL4787900)
Affinity DataIC50: 299nMAssay Description:Binding affinity to human integrin alphaVbeta6 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565936(CHEMBL4799980)
Affinity DataIC50: 311nMAssay Description:Binding affinity to human integrin alphaVbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565945(CHEMBL4795994)
Affinity DataIC50: 471nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565934(CHEMBL4791029)
Affinity DataIC50: 472nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565942(CHEMBL4790959)
Affinity DataIC50: 610nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-8(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565946(CHEMBL4787900)
Affinity DataIC50: 1.01E+3nMAssay Description:Binding affinity to human integrin alphaVbeta8 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565946(CHEMBL4787900)
Affinity DataIC50: 2.08E+3nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565942(CHEMBL4790959)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human integrin alpha2bbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565943(CHEMBL4787559)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human integrin alpha2bbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565944(CHEMBL4793182)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human integrin alpha2bbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565945(CHEMBL4795994)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human integrin alpha2bbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565946(CHEMBL4787900)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human integrin alpha2bbeta3 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetIntegrin alpha-5/beta-1(Human)
Bielefeld University

Curated by ChEMBL
LigandPNGBDBM50565936(CHEMBL4799980)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human integrin alpha5beta1 incubated for 1 hr by ELISA based solid phase integrin binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed