Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50013115
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562736(CHEMBL4752329)
Affinity DataIC50: 0.460nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562729(CHEMBL4748265)
Affinity DataIC50: 0.520nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562734(CHEMBL4763867)
Affinity DataIC50: 0.740nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562727(CHEMBL4744905)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50214615(CHEBI:64177 | Clobenpropit)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562735(CHEMBL4753961)
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562732(CHEMBL4740932)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562728(CHEMBL4741097)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562733(CHEMBL4790392)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562726(CHEMBL4764747)
Affinity DataIC50: 4.30nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562722(CHEMBL4790750)
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562721(CHEMBL4746962)
Affinity DataIC50: 6.5nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562730(CHEMBL4742309)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562731(CHEMBL4789311)
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562742(CHEMBL4751577)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562741(CHEMBL4753396)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562739(CHEMBL4748967)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562738(CHEMBL4749796)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562723(CHEMBL4765168)
Affinity DataIC50: 108nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562724(CHEMBL4742244)
Affinity DataIC50: 167nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562737(CHEMBL4764966)
Affinity DataIC50: 351nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562740(CHEMBL4782278)
Affinity DataIC50: 385nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H3 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562725(CHEMBL4750326)
Affinity DataIC50: 1.79E+3nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H1 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562729(CHEMBL4748265)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human histamine H1 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H2 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562729(CHEMBL4748265)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human histamine H2 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistamine H4 receptor(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50562729(CHEMBL4748265)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human histamine H4 receptor expressed in HEK293 cells preincubated for 5 mins followed by forskolin-stimulation and measured a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed