Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50012374
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chongqing Medical University
Curated by ChEMBL
Chongqing Medical University
Curated by ChEMBL
Affinity DataEC50: 900nMAssay Description:Partial agonist activity at full length human PPARG expressed in African green monkey COS7 cells assessed as increase in receptor activation incubate...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chongqing Medical University
Curated by ChEMBL
Chongqing Medical University
Curated by ChEMBL
Affinity DataEC50: 7.60E+3nMAssay Description:Partial agonist activity at full length human PPARG expressed in African green monkey COS7 cells assessed as increase in receptor activation incubate...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chongqing Medical University
Curated by ChEMBL
Chongqing Medical University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to GST-tagged PPARG LBD (unknown origin) by Fluormone Pan-PPAR Green tracer based TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chongqing Medical University
Curated by ChEMBL
Chongqing Medical University
Curated by ChEMBL
Affinity DataKi: 8.90E+3nMAssay Description:Binding affinity to GST-tagged PPARG LBD (unknown origin) by Fluormone Pan-PPAR Green tracer based TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
Chongqing Medical University
Curated by ChEMBL
Chongqing Medical University
Curated by ChEMBL
Affinity DataKi: 2.20E+4nMAssay Description:Binding affinity to GST-tagged PPARG LBD (unknown origin) by Fluormone Pan-PPAR Green tracer based TR-FRET assayMore data for this Ligand-Target Pair
