Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50048777
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227340(CHEMBL27155)
Affinity DataKi:  48nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50021453(CHEMBL156627 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-t...)
Affinity DataKi:  54nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227341(CHEMBL347866)
Affinity DataKi:  77nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227338(CHEMBL157856)
Affinity DataKi:  140nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  140nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50021448(8-(2-Hydroxy-4-methoxy-phenyl)-1,3-dipropyl-3,7-di...)
Affinity DataKi:  180nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50007838(CHEMBL160369 | 8-Cyclohexyl-1,3-dipropyl-3,7-dihyd...)
Affinity DataKi:  190nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227335(CHEMBL345595)
Affinity DataKi:  240nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50018151(4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-pu...)
Affinity DataKi:  320nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50021449(8-(2,4-Dihydroxy-phenyl)-1,3-dipropyl-3,9-dihydro-...)
Affinity DataKi:  820nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227339(CHEMBL158077)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50007840(8-Cyclopentylmethyl-1,3-dipropyl-3,9-dihydro-purin...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50023353([4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-p...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227332(CHEMBL158507)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227333(CHEMBL346126)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50004568(8-Cyclohexylmethyl-1,3-dipropyl-3,9-dihydro-purine...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50021455(8-(4-Methoxy-phenyl)-1,3-dipropyl-3,9-dihydro-puri...)
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50023354(1,3-Dipropyl-8-pyrazin-2-yl-3,9-dihydro-purine-2,6...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227336(CHEMBL156055)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227334(CHEMBL155951)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227342(CHEMBL155791)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
National Institute of Diabetes, Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50227331(CHEMBL157655)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibition of 5'-(N-ethylcarbamoyl)adenosine-elicited stimulation of adenylate cyclase in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/1/2019
Entry Details Article
PubMed