Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50012013
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553240(CHEMBL4798970)
Affinity DataKi:  33nMAssay Description:Competitive inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by substrate addition and...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 48nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553240(CHEMBL4798970)
Affinity DataIC50: 60nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553241(CHEMBL4752653)
Affinity DataIC50: 241nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553239(CHEMBL4752462)
Affinity DataIC50: 336nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553243(CHEMBL4779124)
Affinity DataIC50: 502nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553242(CHEMBL4741381)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553244(CHEMBL4778612)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM50553245(CHEMBL4793973)
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Anadolu University

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataIC50: 4.66E+3nMAssay Description:Inhibition of human recombinant MAO-A using tyramine as substrate preincubated with enzyme for 30 mins followed by incubation with substrate for 30 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed