Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50013137
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562969(CHEMBL4758943)
Affinity DataKd:  3.40E+3nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant in presence of 0.5% DMSO by surface plasmon resonance analys...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562970(CHEMBL4762702)
Affinity DataKd:  5.70E+3nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562966(CHEMBL4747788)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562969(CHEMBL4758943)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562971(CHEMBL4797205)
Affinity DataKd:  8.90E+3nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by isothermal titration calorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562969(CHEMBL4758943)
Affinity DataIC50: 1.73E+4nMAssay Description:Displacement of Halo-tagged Histone H3.3 from Nanoluc-tagged NSD2- PWWP1 (unknown origin) transfected in human U2OS cells preincubated for one day fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562971(CHEMBL4797205)
Affinity DataKd:  4.10E+4nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562967(CHEMBL4742287)
Affinity DataKd:  7.40E+4nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562959(CHEMBL4752461)
Affinity DataKd:  1.10E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562968(CHEMBL4780499)
Affinity DataKd:  1.14E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562962(CHEMBL4739882)
Affinity DataKd:  1.38E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562961(CHEMBL4756612)
Affinity DataKd:  1.60E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562964(CHEMBL4747137)
Affinity DataKd:  1.73E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562958(CHEMBL4785465)
Affinity DataKd:  1.75E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562963(CHEMBL4789766)
Affinity DataKd:  1.78E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562960(CHEMBL4756809)
Affinity DataKd:  2.08E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHistone-lysine N-methyltransferase NSD2(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50562965(CHEMBL4755270)
Affinity DataKd:  2.97E+5nMAssay Description:Binding affinity to NSD2 PWWP1 domain (unknown origin) assessed as dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed