Compile Data Set for Download or QSAR
Report error Found 59 Enz. Inhib. hit(s) with all data for entry = 50013156
TargetRelaxin receptor 1(Rat)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563220(CHEMBL4793799)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563189(CHEMBL4748830)
Affinity DataEC50:  45nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563219(CHEMBL4797258)
Affinity DataEC50:  18nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563220(CHEMBL4793799)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563221(CHEMBL4752287)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563222(CHEMBL4797641)
Affinity DataEC50:  1nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563223(CHEMBL4799907)
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563224(CHEMBL4764326)
Affinity DataEC50:  1nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563225(CHEMBL4795810)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563226(CHEMBL4745611)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563227(CHEMBL4786789)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563228(CHEMBL4796713)
Affinity DataEC50:  809nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563229(CHEMBL4746080)
Affinity DataEC50:  368nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataEC50:  0.420nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Rat)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563215(CHEMBL4781560)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563218(CHEMBL4744987)
Affinity DataEC50:  18nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Rat)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at rat RXFP1 expressed in human HEK296 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX for 40 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563219(CHEMBL4797258)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563220(CHEMBL4793799)
Affinity DataEC50:  270nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563222(CHEMBL4797641)
Affinity DataEC50:  31nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563223(CHEMBL4799907)
Affinity DataEC50:  9nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563224(CHEMBL4764326)
Affinity DataEC50:  87nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563225(CHEMBL4795810)
Affinity DataEC50:  18nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563226(CHEMBL4745611)
Affinity DataEC50:  20nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563227(CHEMBL4786789)
Affinity DataEC50:  25nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563228(CHEMBL4796713)
Affinity DataEC50: >2.00E+3nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563229(CHEMBL4746080)
Affinity DataEC50: >2.00E+3nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563231(CHEMBL4780098)
Affinity DataEC50:  7.59E+3nMAssay Description:Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563230(CHEMBL4754949)
Affinity DataEC50:  0.0324nMAssay Description:Agonist activity at human RXFP1 expressed in human HEK-293T cells co-transfected with pCRE beta-galactosidase reporter plasmid assessed as inhibition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563202(CHEMBL4761424)
Affinity DataEC50:  200nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563190(CHEMBL4757578)
Affinity DataEC50:  143nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563191(CHEMBL4748931)
Affinity DataEC50:  20nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563192(CHEMBL4800116)
Affinity DataEC50:  146nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563193(CHEMBL4743958)
Affinity DataEC50:  393nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563194(CHEMBL4754697)
Affinity DataEC50:  522nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563195(CHEMBL4747756)
Affinity DataEC50:  124nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563196(CHEMBL4791290)
Affinity DataEC50:  32nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563197(CHEMBL4744303)
Affinity DataEC50:  498nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563198(CHEMBL4743539)
Affinity DataEC50:  17nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563199(CHEMBL4756139)
Affinity DataEC50:  46nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563200(CHEMBL4792874)
Affinity DataEC50:  202nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563201(CHEMBL4781482)
Affinity DataEC50:  929nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563217(CHEMBL4781139)
Affinity DataEC50:  45nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563203(CHEMBL4765167)
Affinity DataEC50:  897nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563204(CHEMBL4791486)
Affinity DataEC50:  54nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563205(CHEMBL4785899)
Affinity DataEC50:  92nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563206(CHEMBL4757890)
Affinity DataEC50:  708nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563207(CHEMBL4755289)
Affinity DataEC50:  230nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563208(CHEMBL4748601)
Affinity DataEC50:  37nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetRelaxin receptor 1(Human)
Sanofi R&D

Curated by ChEMBL
LigandPNGBDBM50563209(CHEMBL4777259)
Affinity DataEC50:  17nMAssay Description:Agonist activity at RXFP1 endogenously expressed in human OVCAR-5 cells assessed as increase in IBMX-induced cAMP accumulation pretreated with IBMX f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Displayed 1 to 50 (of 59 total ) | Next | Last >>
Jump to: