Compile Data Set for Download or QSAR
Report error Found 300 Enz. Inhib. hit(s) with all data for entry = 50013198
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563555(CHEMBL4750420)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase-like 3(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM31085(cid_11409972 | 1-[4-[(4-ethylpiperazin-1-yl)methyl...)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of CDKL3 (unknown origin) by NanoBRET cellular target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50560704(CHEMBL4754195)
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant CLK1 using ERMRPRKRQGSVR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MLK1 (unknown origin) by NanoBRET cellular target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50560704(CHEMBL4754195)
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563539(CHEMBL4762964)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant CLK1 using ERMRPRKRQGSVR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563539(CHEMBL4762964)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563556(CHEMBL4743939)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563537(CHEMBL4789951)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CLK1 using ERMRPRKRQGSVR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563538(CHEMBL4797457)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563539(CHEMBL4762964)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563555(CHEMBL4750420)
Affinity DataIC50: 16nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563538(CHEMBL4797457)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563538(CHEMBL4797457)
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant CLK1 using ERMRPRKRQGSVR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563537(CHEMBL4789951)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50560704(CHEMBL4754195)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563555(CHEMBL4750420)
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50560704(CHEMBL4754195)
Affinity DataIC50: 29nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563539(CHEMBL4762964)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563555(CHEMBL4750420)
Affinity DataIC50: 31nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563556(CHEMBL4743939)
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563537(CHEMBL4789951)
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 3(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563555(CHEMBL4750420)
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563556(CHEMBL4743939)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 39nMAssay Description:Inhibition of MLK3 (unknown origin) by NanoBRET cellular target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563541(CHEMBL4743730)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563554(CHEMBL4790030)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563541(CHEMBL4743730)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563541(CHEMBL4743730)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563554(CHEMBL4790030)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563557(CHEMBL4790791)
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563556(CHEMBL4743939)
Affinity DataIC50: 46nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563541(CHEMBL4743730)
Affinity DataIC50: 51nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563535(CHEMBL4791451)
Affinity DataIC50: 52nMAssay Description:Inhibition of human recombinant CLK4 using YRRAAVPPSPSLS substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563535(CHEMBL4791451)
Affinity DataIC50: 59nMAssay Description:Inhibition of human recombinant CLK1 using ERMRPRKRQGSVR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563554(CHEMBL4790030)
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant HIPK1 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 3(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563541(CHEMBL4743730)
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 3(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563556(CHEMBL4743939)
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563541(CHEMBL4743730)
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant CLK1 using ERMRPRKRQGSVR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563540(CHEMBL4740998)
Affinity DataIC50: 68nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563538(CHEMBL4797457)
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant HIPK2 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563554(CHEMBL4790030)
Affinity DataIC50: 72nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563559(CHEMBL4587433)
Affinity DataIC50: 74nMAssay Description:Inhibition of HIPK2 (unknown origin) by selectscreen kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50563535(CHEMBL4791451)
Affinity DataIC50: 90nMAssay Description:Inhibition of human recombinant CLK2 using YRRAAVPPSPSLSR substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM17055((9S)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydr...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 1(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50242737((R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimet...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetHomeodomain-interacting protein kinase 2(Human)
Masaryk University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Displayed 1 to 50 (of 300 total ) | Next | Last >>
Jump to: