Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50013865
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570416(CHEMBL4871403)
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human APJ receptor stably expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567169(CHEMBL4873876)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at human APJ receptor stably expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567169(CHEMBL4873876)
Affinity DataEC50:  0.0240nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570426(CHEMBL4876050)
Affinity DataEC50:  0.580nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570425(CHEMBL4866313)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570424(CHEMBL4860991)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570423(CHEMBL4846150)
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570422(CHEMBL4852391)
Affinity DataEC50:  15nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570421(CHEMBL4878068)
Affinity DataEC50:  450nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570420(CHEMBL4861053)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570419(CHEMBL4861906)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570418(CHEMBL4857233)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570417(CHEMBL4858384)
Affinity DataEC50:  31nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570414(CHEMBL4861181)
Affinity DataEC50:  450nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570421(CHEMBL4878068)
Affinity DataEC50:  180nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570415(CHEMBL4873340)
Affinity DataEC50:  330nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570416(CHEMBL4871403)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570417(CHEMBL4858384)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570418(CHEMBL4857233)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570419(CHEMBL4861906)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570420(CHEMBL4861053)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570415(CHEMBL4873340)
Affinity DataEC50:  430nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570422(CHEMBL4852391)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570423(CHEMBL4846150)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570424(CHEMBL4860991)
Affinity DataEC50:  0.940nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570425(CHEMBL4866313)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570426(CHEMBL4876050)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567169(CHEMBL4873876)
Affinity DataEC50:  0.0230nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570414(CHEMBL4861181)
Affinity DataEC50:  980nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567169(CHEMBL4873876)
Affinity DataKi:  0.0740nMAssay Description:Displacement of [3H]Apelin-13 from human APJ receptor stably expressed in human HEK293 cell membrane incubated for 120 mins by TopCount scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Bristol Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]Apelin-13 from human APJ receptor stably expressed in human HEK293 cell membrane incubated for 120 mins by TopCount scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed