Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50018393
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of human PHGDH expressed in Escherichia coli BL21 using 3-PG as substrate incubated for 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 9.76E+3nMAssay Description:Inhibition of human PHGDH expressed in Escherichia coli BL21 using 3-PG as substrate incubated for 30 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKd: 1.52E+4nMAssay Description:Binding affinity to human PHGDH expressed in Escherichia coli BL21 incubated for 30 mins by MST assayMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.16E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 2.81E+4nMAssay Description:Inhibition of human full-length PHGDH incubated for 10 mins by SPR analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.48E+4nMAssay Description:Inhibition of human full-length PHGDH incubated for 10 mins by SPR analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.57E+4nMAssay Description:Inhibition of human full-length PHGDH incubated for 10 mins by SPR analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 3.64E+4nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of human full-length PHGDH incubated for 10 mins by SPR analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 4.59E+4nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 6.73E+4nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PHGDH using 3-PG as substrate incubated for 60 mins by fluorescence based analysisMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataKd: 4.70E+5nMAssay Description:Binding affinity to PHGDH (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetD-3-phosphoglycerate dehydrogenase(Human)
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Shanghai University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human PHGDH by fluorescence based analysisMore data for this Ligand-Target Pair

































3D Structure (crystal)














